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ZLD1039 is a potent, highly selective, and orally bioavailable EZH2 inhibitor. ZLD1039 shows potent and concentration-dependent inhibition of PRC2 enzymatic activity against EZH2 wild-type as well as Y641F, and A677G mutant enzymes with IC50 values of 5.6, 15, and 4.0 nM, respectively. ZLD1039 inhibits breast tumor growth and metastasis.
| Molecular Weight | 612.8 |
| Formula | C36H48N6O3 |
| CAS Number | 1826865-46-6 |
| Form | Solid |
| Solubility (25°C) | DMSO 9.09 mg/mL (ultrasonic and adjust pH to 3 with 1M HCl) |
| Storage | 4°C, protect from light |
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