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WHI-P258

Cat. No. M10695

All AbMole products are for research use only, cannot be used for human consumption.

WHI-P258  Structure
Size Price Availability Quantity
5mg USD 65 In stock
10mg USD 95 In stock
25mg USD 215 In stock
50mg USD 380 In stock
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Quality Control & Documentation
Biological Activity

WHI-P258 is an inhibitor of JAK3 with a Ki value of 72 μM.

Chemical Information
Molecular Weight 281.31
Formula C16H15N3O2
CAS Number 21561-09-1
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] E A Sudbeck, et al. Clin Cancer Res. Structure-based design of specific inhibitors of Janus kinase 3 as apoptosis-inducing antileukemic agents

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Keywords: WHI-P258 supplier, JNK, inhibitors, activators

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