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WH-4-023

Cat. No. M3676

All AbMole products are for research use only, cannot be used for human consumption.

WH-4-023 Structure
Synonym:

Dual LCK/SRC inhibitor

Size Price Availability Quantity
Free Sample (0.5-1 mg)  USD 0 In stock
10mM*1mL in DMSO USD 80 In stock
2mg USD 36 In stock
5mg USD 60 In stock
10mg USD 100 In stock
50mg USD 220 In stock
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Quality Control & Documentation
Biological Activity

WH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM. WH-4-023 has little inhibition on p38α and KDR.

Chemical Information
Molecular Weight 568.67
Formula C32H36N6O4
CAS Number 837422-57-8
Solubility (25°C) DMSO 15 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Martin MW, et al. J Med Chem. Novel 2-aminopyrimidine carbamates as potent and orally active inhibitors of Lck: synthesis, SAR, and in vivo antiinflammatory activity.

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  Catalog
Abmole Inhibitor Catalog




Keywords: WH-4-023, Dual LCK/SRC inhibitor supplier, Src-bcr-Abl, inhibitors, activators

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