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VU0453379 

Cat. No. M28746

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VU0453379  Structure

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Quality Control & Documentation
Biological Activity

VU0453379 is a highly selective and central nervous system (CNS) penetrant positive allosteric modulator (PAM) of glucagon-like peptide-1R (GLP-1R) with an EC50 of 1.3 μM.

Chemical Information
Molecular Weight 434.57
Formula C26H34N4O2
CAS Number 1638646-27-1
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Lindsey C Morris, et al. J Med Chem. Discovery of (S)-2-cyclopentyl-N-((1-isopropylpyrrolidin2-yl)-9-methyl-1-oxo-2,9-dihydro-1H-pyrrido[3,4-b]indole-4-carboxamide (VU0453379): a novel, CNS penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM)

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  Catalog
Abmole Inhibitor Catalog




Keywords: VU0453379  supplier, GLP Receptor, inhibitors, activators

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