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Velusetrag (TD-5108) hydrochloride is an orally active, potent and selective agonist of serotonin 5-HT4 receptor (5-HT4R), with a pKi of 7.7. Velusetrag hydrochloride exhibits no affinity (Ki>10 μM) for 5-HT2A and 5-HT2B receptors. Velusetrag hydrochloride can be used for the research of gastrointestinal diseases and Parkinson's disease.
| Molecular Weight | 541.1 |
| Formula | C25H37ClN4O5S |
| CAS Number | 866933-51-9 |
| Form | Solid |
| Solubility (25°C) | DMSO 220 mg/mL (ultrasonic) Water 10 mg/mL (ultrasonic and warming and heat to 60°C) |
| Storage | 4°C, dry, sealed |
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