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UNP-6457

Cat. No. M41352

All AbMole products are for research use only, cannot be used for human consumption.

UNP-6457 Structure

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Quality Control & Documentation
Biological Activity

UNP-6457 is a potent active MDM2-p53 interaction inhibitor with an IC50 values of 8.9 nM.

Chemical Information
Molecular Weight 1229.31
Formula C62H71F3N14O10
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Anthony P Silvestri et al. ACS Med Chem Lett. DNA-Encoded Macrocyclic Peptide Libraries Enable the Discovery of a Neutral MDM2-p53 Inhibitor

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NSC 66811

NSC 66811 is a potent MDM2 inhibitor with Ki value of 120 nM, which disrupts MDM2-p53 interaction and activates p53 function.

Nutlin-3a

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SL-01

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  Catalog
Abmole Inhibitor Catalog




Keywords: UNP-6457 supplier, Mdm2, inhibitors, activators

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