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Unecritinib

Cat. No. M45163

All AbMole products are for research use only, cannot be used for human consumption.

Unecritinib Structure
Synonym:

TQ-B3101

Size Price Availability Quantity
1mg USD 300 In stock
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Quality Control & Documentation
Biological Activity

Unecritinib is a potent EGFR tyrosine kinase inhibitor that inhibits ALK, ROS1, and MET and has anticancer activity. Unecritinib is indicated for use in studies of solid tumors and ALK-positive anaplastic large cell lymphoma.

Chemical Information
Molecular Weight 492.37
Formula C23H24Cl2FN5O2
CAS Number 1418026-92-2
Solubility (25°C) DMSO 100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hong Wang, et al. J Pharm Biomed Anal. Simultaneous determination of unecritinib (TQ-B3101) and its active metabolite crizotinib in rat plasma by LC-MS/MS:An application to pharmacokinetic studies

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Keywords: Unecritinib, TQ-B3101 supplier, EGFR/HER2, inhibitors, activators

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