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Umbralisib hydrochloride (TGR-1202 hydrochloride) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Umbralisib hydrochloride (TGR-1202 hydrochloride) is also active against CK1ε, with an EC50 value of 6.0 μM.
| Molecular Weight | 608.01 |
| CAS Number | 1532533-78-0 |
| Solubility (25°C) | DMSO ≥ 100 mg/mL |
| Storage | 2-8°C, dry, sealed |
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