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Tyrphostin AG528

Cat. No. M9722

All AbMole products are for research use only, cannot be used for human consumption.

Tyrphostin AG528 Structure
Synonym:

Tyrphostin B66; AG-528

Size Price Availability Quantity
5mg USD 45 In stock
10mg USD 85 In stock
25mg USD 155 In stock
50mg USD 270 In stock
100mg USD 480 In stock
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Quality Control & Documentation
Biological Activity

Tyrphostin AG528 (Tyrphostin B66) is an inhibitor of EGFR and ErbB2 with IC50 values of 4.9 and 2.1 μM, respectively. The natural bond orbital (NBO) analysis suggested that the molecule Tyrphostin AG528 as an electron donor and the CNT(6,6-6) nanotube play the role of an electron acceptor at the complex CNT(6,6-6)/Tyrphostin AG528.

Chemical Information
Molecular Weight 306.32
Formula C18H14N2O3
CAS Number 133550-49-9
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Masoome Sheikhi, et al. Curr Mol Med. Investigation of Adsorption Tyrphostin AG528 Anticancer Drvg Upon the CNT(6,6-6) Nanotube: A DFT Study

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Abmole Inhibitor Catalog




Keywords: Tyrphostin AG528, Tyrphostin B66; AG-528 supplier, EGFR/HER2, inhibitors, activators

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