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TRIM24/BRPF1-IN-2

Cat. No. M41649

All AbMole products are for research use only, cannot be used for human consumption.

TRIM24/BRPF1-IN-2 Structure

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Quality Control & Documentation
Biological Activity

TRIM24/BRPF1-IN-2 is a potent TRIM24/BRPF1 dual inhibitor, with IC50 values of 0.98 and 1.16 μM, respectively.

Chemical Information
Molecular Weight 386.46
Formula C20H22N2O4S
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Tingting Jiang et al. Acta Pharm Sin B. Development of small-molecule tropomyosin receptor kinase (TRK) inhibitors for NTRK fusion cancers

[2] Hui Zhang et al. Cancer Res. Deregulation of SPOP in Cancer

[3] Shigetsugu Hatakeyama. Nat Rev Cancer. TRIM proteins and cancer

[4] Monisankar Ghosh et al. Mol Cell. p53 engages the cGAS/STING cytosolic DNA sensing pathway for tumor suppression

[5] Seung Koo Yang et al. Allergy Asthma Immunol Res. The Role of TRIM24 in Allergic Rhinitis

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  Catalog
Abmole Inhibitor Catalog




Keywords: TRIM24/BRPF1-IN-2 supplier, Epigenetic Reader Domain, inhibitors, activators

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