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TPOP146

Cat. No. M13826

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TPOP146 Structure

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Quality Control & Documentation
Biological Activity

TPOP146 is a selective CBP/P300 benzoxazepine bromodomain inhibitor with Kd values of 134 nM and 5.02 μM for CBP and BRD4.

Chemical Information
Molecular Weight 481.58
CAS Number 2018300-62-2
Solubility (25°C) DMSO ≥ 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Tobias A Popp, et al. J Med Chem. Development of Selective CBP/P300 Benzoxazepine Bromodomain Inhibitors

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  Catalog
Abmole Inhibitor Catalog




Keywords: TPOP146 supplier, Epigenetic Reader Domain, inhibitors, activators

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