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TP-238 is a potent and selective dual CECR2/BPTF probe with IC50 values of 30 nM and 350 nM, respectively. TP-238 also inhibits BRD9 with a pIC50 of 5.9 and is less active against other 338 kinases.
| Molecular Weight | 458.58 |
| Formula | C22H30N6O3S |
| CAS Number | 2415263-04-4 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[1] Tian Lu, et al. J Med Chem. Discovery of High-Affinity Inhibitors of the BPTF Bromodomain
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