All AbMole products are for research use only, cannot be used for human consumption.
Tivumecirnon is a potent CCR4 small molecule antagonist with antitumor activity that blocks regulatory T cells that interfere with an effective antitumor immune response. It can be used in melanoma related studies.
| Molecular Weight | 543.41 |
| Formula | C24H27Cl2F3N6O |
| CAS Number | 2174938-78-2 |
| Form | Solid |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related CCR Products |
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| Vicriviroc Malate
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| Bindarit
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| BMS-813160
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| INCB3284 dimesylate
INCB 3284 dimesylate is a potent, selective and orally bioavailable hCCR2 antagonist with IC50 of 3.7 nM. |
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