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THK01

Cat. No. M41592

All AbMole products are for research use only, cannot be used for human consumption.

THK01 Structure

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Quality Control & Documentation
Biological Activity

THK01 is a potent ROCK2 inhibitor with IC50 values of 5.7 and 923 nM for ROCK2 and ROCK1, respectively.

Chemical Information
Molecular Weight 327.34
Formula C20H13N3O2
CAS Number 2226941-26-8
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jinhui Wang et al. Eur J Med Chem. Discovery of unglycosylated indolocarbazoles as ROCK2 isoform-selective inhibitors for the treatment of breast cancer metastasis

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  Catalog
Abmole Inhibitor Catalog




Keywords: THK01 supplier, ROCK, inhibitors, activators

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