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Thiethylperazine dimaleate, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Thiethylperazine dimaleate is also a selective ABCC1activator that reduces amyloid-β (Aβ) load in mice. Thiethylperazine dimaleate has anti-emetic, antipsychotic and antimicrobial effects.
| Molecular Weight | 631.76 |
| Formula | C30H37N3O8S2 |
| CAS Number | 1179-69-7 |
| Form | Solid |
| Solubility (25°C) | DMSO 125 mg/mL (ultrasonic and warming and heat to 60°C) |
| Storage | 4°C, protect from light, dry, sealed |
[3] M Tsuru, et al. No To Shinkei. [Clinical experiences with thiethylperazine dimaleate (Toresten)]
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