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TC NTR1 17

Cat. No. M7362

All AbMole products are for research use only, cannot be used for human consumption.

TC NTR1 17 Structure

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Quality Control & Documentation
Biological Activity

TC NTR1 17 is a non-peptide neurotensin receptor 1 (NTS1) partial agonist (EC50 <15.6 nM and Emax = 63% of neurotensin response in Ca2+ mobilization assay). Exhibits over 50-fold selectivity for NTS1 over NTS2 and GPR35.

Chemical Information
Molecular Weight 522.98
Formula C27H27ClN4O5
CAS Number 1146757-96-1
Solubility (25°C) 1eq. NaOH 26.15 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Bohm, et al. Biochem J. Molecular cloning, expression and potential functions of the human proteinase-activated receptor-2.

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Keywords: TC NTR1 17 supplier, inhibitors, activators

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