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Taprenepag

Cat. No. M9854

All AbMole products are for research use only, cannot be used for human consumption.

Taprenepag Structure
Synonym:

CP-544326

Size Price Availability Quantity
5mg USD 75 In stock
10mg USD 120 In stock
25mg USD 250 In stock
50mg USD 400 In stock
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Quality Control & Documentation
Biological Activity

Taprenepag (CP-544326) is a potent selective prostagenin EP(2) agonist with IC50 of 10 and 15 nM for human and rat EP2, respectively. Taprenepag has higher selectivity for EP2 than other EP receptors (IC50>3200 nM for EP1, EP3 and EP4) and a group of 37 G-protein-coupled receptors.

Chemical Information
Molecular Weight 478.52
Formula C24H22N4O5S
CAS Number 752187-80-7
Solubility (25°C) DMSO 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Ganesh Prasanna, et al. Exp Eye Res. Effect of PF-04217329 a prodrug of a selective prostaglandin EP(2) agonist on intraocular pressure in preclinical models of glaucoma

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Keywords: Taprenepag, CP-544326 supplier, Prostaglandin Receptor, inhibitors, activators

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