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Src interactivator-1 is a highly selective, ATP-competitive, two-site Src tyrosine kinase Inhibitor with IC50 values of 44 nM and 88 nM against Src and Lck, respectively. Src interactivator-1 also inhibits Csk and Yes.
| Molecular Weight | 373.4 |
| Formula | C22H19N3O3 |
| CAS Number | 179248-59-0 |
| Form | Solid |
| Solubility (25°C) | DMSO: ≥10 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[4] Stephen P Higgins, et al. TGF-β1/p53 signaling in renal fibrogenesis
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