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SR-4133

Cat. No. M41416

All AbMole products are for research use only, cannot be used for human consumption.

SR-4133 Structure

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Quality Control & Documentation
Biological Activity

SR-4133 is a potent and highly CK1ε selective inhibitor with an IC50 of 58 nM.

Chemical Information
Molecular Weight 512.51
Formula C27H22F2N8O
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jun Yong Choi et al. J Med Chem. Structure-Based Development of Isoform-Selective Inhibitors of Casein Kinase 1ε vs Casein Kinase 1δ

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  Catalog
Abmole Inhibitor Catalog




Keywords: SR-4133 supplier, Casein Kinase, inhibitors, activators

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