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Squarunkin A 

Cat. No. M29235

All AbMole products are for research use only, cannot be used for human consumption.

Squarunkin A  Structure

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Quality Control & Documentation
Biological Activity

Squarunkin A is a potent and selective UNC119-cargo interaction inhibitor, interrupting the UNC119A-myristoylated Src N-terminal peptide interaction (IC50=10 nM). Squarunkin A interferes with the activation of Src kinase in cells.

Chemical Information
Molecular Weight 523.55
Formula C25H32F3N5O4
CAS Number 2101958-02-3
Form Solid
Solubility (25°C) DMSO 9.62 mg/mL (ultrasonic and warming and heat to 60°C)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Tom Mejuch, et al. Angew Chem Int Ed Engl. Small-Molecule Inhibition of the UNC119-Cargo Interaction

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  Catalog
Abmole Inhibitor Catalog




Keywords: Squarunkin A  supplier, Src-bcr-Abl, inhibitors, activators

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