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SHR168442

Cat. No. M21134

All AbMole products are for research use only, cannot be used for human consumption.

SHR168442 Structure

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Quality Control & Documentation
Biological Activity

SHR168442 is a modulator of RORγ with an IC50 value of 0.035 μM. It can be used as a skin-restricted topical compound for the study of psoriasis.

Chemical Information
Molecular Weight 532.43
Formula C23H25Cl2F2N3O3S
CAS Number 2382961-86-4
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Suxing Liu, et al. Sci Rep. Discovery of a novel RORγ antagonist with skin-restricted exposure for topical treatment of mild to moderate psoriasis

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  Catalog
Abmole Inhibitor Catalog




Keywords: SHR168442 supplier, ROR, inhibitors, activators

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