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SB-423557 

Cat. No. M29964

All AbMole products are for research use only, cannot be used for human consumption.

SB-423557  Structure

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Quality Control & Documentation
Biological Activity

SB-423557 is an orally active calcium-sensing receptor (CaR) antagonist (IC50=520 nM), precursor of SB-423562 (IC50=73 nM). SB-423557 is well tolerated in human and increases plasma concentrations of exogenous parathyroid hormone (PTH) and stimulates bone formation.

Chemical Information
Molecular Weight 464.6
Formula C28H36N2O4
CAS Number 351490-26-1
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Sanjay Kumar, et al. Bone. An orally active calcium-sensing receptor antagonist that transiently increases plasma concentrations of PTH and stimulates bone formation

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  Catalog
Abmole Inhibitor Catalog




Keywords: SB-423557  supplier, Calcium-sensing Receptor, inhibitors, activators

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