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SB-277011 dihydrochloride

Cat. No. M27982

All AbMole products are for research use only, cannot be used for human consumption.

SB-277011 dihydrochloride Structure
Synonym:

SB-277011A dihydrochloride

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Quality Control & Documentation
Biological Activity

SB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively.

Chemical Information
Molecular Weight 511.49
Formula C28H32Cl2N4O
CAS Number 1226917-67-4
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Béla Kiss, et al. Naunyn Schmiedebergs Arch Pharmacol. Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

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Keywords: SB-277011 dihydrochloride, SB-277011A dihydrochloride supplier, Dopamine Receptor, inhibitors, activators

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