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Sampatrilat (UK-81252) is a potent and orally active vasopeptidase inhibitor of ACE and neutral endopeptidase (NEP). Sampatrilat inhibits C-domain ACE (Ki=13.8 nM) 12.4-fold more potent than that for the N-domain (Ki=171.9 nM). Sampatrilat (UK-81252) can be used for the study of chronic heart failure and blood pressure regulation.
| Molecular Weight | 584.68 |
| Formula | C26H40N4O9S |
| CAS Number | 129981-36-8 |
| Solubility (25°C) | DMSO 100 mg/mL (ultrasonic) |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
[4] Kristina Allikmets. Curr Opin Investig Drugs. Sampatrilat Shire
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