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S1R agonist 1 hydrochloride

Cat. No. M42697

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S1R agonist 1 hydrochloride Structure

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Quality Control & Documentation
Biological Activity

S1R agonist 1 hydrochloride is a selective S1R agonist with Kis of 0.93 nM and 72 nM for S1R and S2R, respectively.

Chemical Information
Molecular Weight 331.88
Formula C20H26ClNO
CAS Number 242487-82-7
Form Solid
Storage -20°C, dry, sealed
References

[1] Alba Vera-Zambrano et al. Pharmacol Res. Sigma-1 receptor modulation fine-tunes KV1.5 channels and impacts pulmonary vascular function

[2] Samantha T Reyes et al. Sci Rep. Effects of the sigma-1 receptor agonist blarcamesine in a murine model of fragile X syndrome: neurobehavioral phenotypes and receptor occupancy

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