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RSM-932A (TCD-717) is a specific ChoKα inhibitor with IC50s of 1 and 33 μM for human recombinant ChoKα and ChoKβ enzymes, respectively. RSM-932A acts as the “first in humans” compound targeting ChoKα. RSM-932A is potent in vitro anti-proliferative and in vivo anti-tumoral activity against human xenografts in mice, showing high efficacy with low toxicity profiles.
| Molecular Weight | 877.53 |
| Formula | C46H38Br2Cl2N4 |
| CAS Number | 850807-63-5 |
| Form | Solid |
| Solubility (25°C) | DMSO 16.67 mg/mL (ultrasonic and warming and heat to 60°C) |
| Storage | 4°C, protect from light, dry, sealed |
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