All AbMole products are for research use only, cannot be used for human consumption.
Rociletinib hydrobromide (CO-1686 hydrobromide) is an orally delivered kinase inhibitor that specifically targets the mutant forms of EGFR including T790M, and the Ki values for EGFRL858R/T790M and EGFRWT are 21.5 nM and 303.3 nM, respectively.
| Molecular Weight | 636.46 |
| Formula | C27H29BrF3N7O3 |
| CAS Number | 1446700-26-0 |
| Solubility (25°C) | DMSO ≥ 50 mg/mL |
| Storage | 2-8°C, dry, sealed |
| Related EGFR/HER2 Products |
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| Sapitinib (AZD8931)
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