Free shipping on all orders over $ 500

RET V804M-IN-1 

Cat. No. M49837

All AbMole products are for research use only, cannot be used for human consumption.

RET V804M-IN-1  Structure

Price and Availability

For this product's availability, delivery time and price, please email inquiry@abmole.com directly or click the "Inquiry Now" button below.


Quality Control & Documentation
Biological Activity

RET V804M-IN-1 is a wt-RET -selective inhibitors of RETV804M kinase, with an IC50 of 20 nM.

Chemical Information
Molecular Weight 344.37
Formula C19H16N6O
CAS Number 2414909-94-5
Form Solid
Solubility (25°C) DMSO 100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
Related RET Products
RPI-1

RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.

SPP86

SPP86 is a potent cell permeable inihbitor of RET tyrosine kinase with an IC50 value of 8 nM and with some inhibitory activity at EphA1, FGFR1, Flt4, Lck and Yes.

Pralsetinib

Pralsetinib (BLU-667) is a next generation highly potent, selective RET inhibitor with IC50 of 0.3-0.4 nM for WT RET, RET mutants V804L, V804M, M918T and CCDC6-RET fusion.

Selpercatinib (LOXO-292)

Selpercatinib (LOXO-292) is a first-in-class, highly selective and potent small molecule RET inhibitor with good blood-brain barrier (BBB) penetration. and RET (G810R) with IC50 values of 14.0 nM, 24.1 nM and 530.7 nM, respectively.

AD80

AD80 is a multikinase inhibitor, it potently targets human RET, BRAF, S6K, and SRC.

  Catalog
Abmole Inhibitor Catalog




Keywords: RET V804M-IN-1  supplier, RET, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2026 AbMole BioScience. All Rights Reserved.