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(rel)-AR234960

Cat. No. M11021

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(rel)-AR234960  Structure

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Quality Control & Documentation
Biological Activity

(rel)-AR234960 is the relatively active configuration of AR234960. AR234960 is a non-peptide MAS (a G protein coupling receptor) agonist that upregulates CTGF mRNA and protein levels through the ERK1/2 signaling pathway in HEK293-MAS cells and adult myocardial fibroblasts.

Chemical Information
Molecular Weight 555.62
Formula C27H30FN5O5S
CAS Number 1408311-94-3
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
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  Catalog
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Keywords: (rel)-AR234960 supplier, ERK, inhibitors, activators

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