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Ralaniten triacetate

Cat. No. M10961

All AbMole products are for research use only, cannot be used for human consumption.

Ralaniten triacetate Structure
Synonym:

EPI-506

Size Price Availability
5mg USD 500 Custom Synthesis
10mg USD 850 Custom Synthesis
25mg USD 1800 Custom Synthesis
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Quality Control & Documentation
Biological Activity

Ralaniten triacetate (EPI-506), a prodrug for Ralaniten, is a pioneering, orally active androgen receptor (AR) N-terminal domain (NTD) inhibitor. Ralaniten triacetate is active against full-length and resistance-related AR species, including AR-v7.

Chemical Information
Molecular Weight 521
Formula C27H33ClO8
CAS Number 1637573-04-6
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jon K Obst, et al. ACS Pharmacol Transl Sci. Revealing Metabolic Liabilities of Ralaniten To Enhance Novel Androgen Receptor Targeted Therapies

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Keywords: Ralaniten triacetate, EPI-506 supplier, Androgen Receptor, inhibitors, activators

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