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(R)-Nepicastat hydrochloride

Cat. No. M2349

All AbMole products are for research use only, cannot be used for human consumption.

(R)-Nepicastat hydrochloride Structure
Synonym:

RS-25560-198 HCl

Size Price Availability
10mg USD 220 Out of stock
50mg USD 550 Out of stock
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Quality Control & Documentation
Biological Activity

Nepicastat is a novel inhibitor of dopamine-beta-hydroxylase, the enzyme which catalyses the conversion of dopamine to noradrenaline in sympathetic nerves. (R)-Nepicastat (30 mg/kg, p.o.) reduces noradrenaline content, dopamine content and dopamine/noradrenaline ratio in mesenteric artery and left ventricle of spontaneously hypertensive rats (SHRs).

Chemical Information
Molecular Weight 331.81
Formula C14H15F2N3S.HCl
CAS Number 195881-94-8
Solubility (25°C) DMSO 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Stanley WC, et al. Br J Pharmacol. Catecholamine modulatory effects of nepicastat (RS-25560-197), a novel, potent and selective inhibitor of dopamine-beta-hydroxylase.

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Keywords: (R)-Nepicastat hydrochloride, RS-25560-198 HCl supplier, HCV Protease, inhibitors, activators

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