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Proxalutamide

Cat. No. M11020

All AbMole products are for research use only, cannot be used for human consumption.

Proxalutamide Structure
Synonym:

GT0918

Size Price Availability Quantity
5mg USD 450 In stock
10mg USD 570 In stock
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Quality Control & Documentation
Biological Activity

Proxalutamide (GT0918) is an antagonist of the androgen receptor (AR) with oral activity. Proxalutamide (GT0918) can be used in prostate cancer and COVID-19 research.

Chemical Information
Molecular Weight 517.50
Formula C₂₄H₁₉F₄N₅O₂S
CAS Number 1398046-21-3
Solubility (25°C) DMSO ≥ 60 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Yue Gu, et al. Int J Mol Sci. Novel Strategy of Proxalutamide for the Treatment of Prostate Cancer through Coordinated Blockade of Lipogenesis and Androgen Receptor Axis

[2] Serap Şimşek-Yavuz, et al. Turk J Med Sci. An update of anti-viral treatment of COVID-19

[3] Hua Sang, et al. Rapid Commun Mass Spectrom. Quantitative determination of proxalutamide in rat plasma and tissues using liquid chromatography/tandem mass spectrometry

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Keywords: Proxalutamide, GT0918 supplier, Androgen Receptor, inhibitors, activators

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