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PNU-177864

Cat. No. M41807

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PNU-177864 Structure

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Quality Control & Documentation
Biological Activity

PNU-177864 is a potent, selective and orally active dopamine D3 receptor antagonist.

Chemical Information
Molecular Weight 402.43
Formula C18H21F3N2O3S
CAS Number 250266-51-4
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Daniel G Rudmann et al. Toxicol Pathol. Epididymal and systemic phospholipidosis in rats and dogs treated with the dopamine D3 selective antagonist PNU-177864

[2] Steven L Vonderfecht et al. Toxicol Pathol. Myopathy related to administration of a cationic amphiphilic drug and the use of multidose drug distribution analysis to predict its occurrence

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Keywords: PNU-177864 supplier, Dopamine Receptor, inhibitors, activators

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