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Pizotifen malate

Cat. No. M2266

All AbMole products are for research use only, cannot be used for human consumption.

Pizotifen malate Structure
Synonym:

Sandomigran, pizotyline

Size Price Availability Quantity
Free Sample (1-2 mg)  USD 0 In stock
50mg USD 30 In stock
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Quality Control & Documentation
Biological Activity

Pizotifen malate is a potent 5-HT2 receptor antagonist, with a high affinity for 5-HT1C binding site. In addition, it has been found to display vasoconstrictor activity in vivo.

Chemical Information
Molecular Weight 429.53
Formula C19H21NS.C4H6O5
CAS Number 5189-11-7
Solubility (25°C) DMSO 35 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Lin OA, et al. PLoS One. The antidepressant 5-HT2A receptor antagonists pizotifen and cyproheptadine inhibit serotonin-enhanced platelet function.

[2] Ujhazy E, et al. Agents Actions. Teratological and cytogenetical evaluation of two antihistamines (pipethiadene and pizotifen maleate) in mice.

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Keywords: Pizotifen malate, Sandomigran, pizotyline supplier, 5-HT Receptor, inhibitors, activators

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