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PF-05241328 

Cat. No. M28305

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PF-05241328  Structure

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Quality Control & Documentation
Biological Activity

PF-05241328 is a potent and selective inhibitor of human Nav1.7 voltage-dependent sodium channels (Nav1.7), with an IC50 of 31 nM.

Chemical Information
Molecular Weight 436.91
Formula C19H21ClN4O4S
CAS Number 1387633-03-5
Form Solid
Solubility (25°C) DMSO 100 mg/mL (ultrasonic and warming and heat to 60°C)
Storage Powder -20°C
References

[1] Hannah M Jones, et al. Clin Pharmacokinet. Clinical Micro-Dose Studies to Explore the Human Pharmacokinetics of Four Selective Inhibitors of Human Nav1.7 Voltage-Dependent Sodium Channels

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  Catalog
Abmole Inhibitor Catalog




Keywords: PF-05241328  supplier, Sodium Channel, inhibitors, activators

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