PF-05105679

Cat. No. M28327

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PF-05105679 is an orally active and selective TRPM8 antagonist with an IC50 of 103 nM. PF-05105679 has the potential for cold-related pain.

Molecular Weight	428.45
Formula	C26H21FN2O3
CAS Number	1398583-31-7
Form	Solid
Solubility (25°C)	DMSO 125 mg/mL (ultrasonic)
Storage	Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month

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