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PETCM

Cat. No. M7112

All AbMole products are for research use only, cannot be used for human consumption.

PETCM Structure
Size Price Availability
5mg USD 50 4-7 Days
10mg USD 80 4-7 Days
50mg USD 240 4-7 Days
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Quality Control & Documentation
Biological Activity

PETCM is a caspase-3 activator. PETCM acts via inhibition of the oncoprotein ProT, therefore stimulates apoptosome formation and subsequent caspase-3 activation in a cytochrome c-dependent manner.

Chemical Information
Molecular Weight 240.51
Formula C8H8Cl3NO
CAS Number 10129-56-3
Solubility (25°C) DMSO ≥ 60 mg/mL (ultrasonic and heat to 40°C)
1eq. HCl: 10 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Terashima, et al. Eur J Pharmacol. R-268712, an orally active transforming growth factor-β type I receptor inhibitor, prevents glomerular sclerosis in a Thy1 nephritis model.

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  Catalog
Abmole Inhibitor Catalog




Keywords: PETCM supplier, Caspase, inhibitors, activators

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