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PD 168368 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15–45 nM. PD 168368 is neuromedin B receptor (NMBR; IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively.
| Molecular Weight | 554.64 |
| Formula | C31H34N6O4 |
| CAS Number | 204066-82-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 30 mg/mL (Need ultrasonic and warming) DMF 10 mg/mL (Need ultrasonic and warming) |
| Storage | Powder -20°C |
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