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PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer.
| Molecular Weight | 272.73 |
| Formula | C15H13ClN2O |
| CAS Number | 2819989-60-9 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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| (+)-JQ1
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