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Fezagepras (Setogepram) sodium acts as an orally active agonist for GPR40 and as an antagonist or inverse agonist for GPR84. Fezagepras sodium decreases renal, liver and pancreatic fibrosis. Fezagepras sodium exerts anti-fibrotic, anti-inflammatory and anti-proliferative actions.
| Molecular Weight | 228.26 |
| Formula | C13H17NaO2 |
| CAS Number | 1254472-97-3 |
| Form | Solid |
| Solubility (25°C) | Water ≥ 100 mg/mL DMSO ≥ 64 mg/mL |
| Storage | 4°C, dry, sealed |
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