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Palazestrant

Cat. No. M45361

All AbMole products are for research use only, cannot be used for human consumption.

Palazestrant Structure
Synonym:

OP-1250

Size Price Availability Quantity
1mg USD 110 In stock
5mg USD 195 In stock
10mg USD 290 In stock
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Quality Control & Documentation
Biological Activity

Palazestrant is a novel, orally active, estrogen receptor antagonist and selective estrogen receptor degrader. It can be used in studies related to ER+/HER2+ breast cancer.

Chemical Information
Molecular Weight 449.60
Formula C28H36FN3O
CAS Number 2092925-89-6
Form Solid
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Walter N Kernan, et al. N Engl J Med. Pioglitazone after Ischemic Stroke or Transient Ischemic Attack

[2] Nathaniel E Margolis, et al. Radiographics. Update on imaging of the postsurgical breast

[3] Sarah Palestrant, et al. Radiol Clin North Am. Approach to breast magnetic resonance imaging interpretation

[4] Marc I Chimowitz, et al. N Engl J Med. Stenting versus aggressive medical therapy for intracranial arterial stenosis

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Keywords: Palazestrant, OP-1250 supplier, Estrogen Receptor, inhibitors, activators

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