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Benzquinamide

Cat. No. M30393

All AbMole products are for research use only, cannot be used for human consumption.

Benzquinamide Structure
Synonym:

P2647; BZQ; Benzoquinamide

Price and Availability

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Quality Control & Documentation
Biological Activity

Benzquinamide (P2647) is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively.

Chemical Information
Molecular Weight 404.5
Formula C22H32N2O5
CAS Number 63-12-7
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] E H WISEMAN, et al. Biochem Pharmacol. THE DISTRIBUTION, EXCRETION AND METABOLISM OF BENZQUINAMIDE

[2] A WEISSMAN, et al. Biochem Pharmacol. Effects of benzquinamide on avoidance behavior and brain amine levels

[3] C G Moertel, et al. Clin Pharmacol Ther. Oral benzquinamide in the treatment of nausea and vomiting

[4] D J Smith, et al. Anesth Analg. Cardiovascular effects of benzquinamide

[5] D C Hobbs, et al. J Pharmacokinet Biopharm. Pharmacokinetics of benzquinamide in man

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Keywords: Benzquinamide, P2647; BZQ; Benzoquinamide supplier, Adrenergic Receptor, inhibitors, activators

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