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OT-R antagonist 1

Cat. No. M29995

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OT-R antagonist 1 Structure
Synonym:

Oxytocin receptor antagonist 1

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Quality Control & Documentation
Biological Activity

OT-R antagonist 1 is a new potent and selective nonpeptide low molecular weight OT-R antagonist. OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM).

Chemical Information
Molecular Weight 471.55
Formula C28H29N3O4
CAS Number 364071-17-0
Form Solid
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hui Huang, et al. Psychopharmacology (Berl). Alcohol-induced conditioned place preference negatively correlates with anxiety-like behavior in adolescent mice: inhibition by a neurokinin-1 receptor antagonist

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Keywords: OT-R antagonist 1, Oxytocin receptor antagonist 1 supplier, Oxytocin Receptor, inhibitors, activators

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