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OM-1700 

Cat. No. M29595

All AbMole products are for research use only, cannot be used for human consumption.

OM-1700  Structure

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Quality Control & Documentation
Biological Activity

OM-1700 is a potent tankyrase inhibitor with IC50s of 127 and 14 nM for tankyrase 1 and tankyrase 2, respectively. OM-1700 reduces cell growth in the colon cancer cell line COLO 320DM (GI50=650 nM).

Chemical Information
Molecular Weight 458.49
Formula C25H23FN6O2
CAS Number 2406276-78-4
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Ruben G G Leenders, et al. J Med Chem. Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II

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  Catalog
Abmole Inhibitor Catalog




Keywords: OM-1700  supplier, PARP, inhibitors, activators

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