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NRX-103094 

Cat. No. M29815

All AbMole products are for research use only, cannot be used for human consumption.

NRX-103094  Structure

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Quality Control & Documentation
Biological Activity

NRX-103094 is a potent enhancer of the interaction between β-catenin, and its cognate E3 ligase, SCFβ-TrCP. NRX-103094 enhances the binding of pSer33/Ser37 β-catenin peptide for β-TrCP with an EC50 of 62 nM and a Kd of 0.6 nM.

Chemical Information
Molecular Weight 503.28
Formula C20H11Cl2F3N2O4S
CAS Number 2763260-36-0
Form Solid
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
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Keywords: NRX-103094  supplier, PROTAC, inhibitors, activators

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