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Naltriben mesylate

Cat. No. M7013

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Naltriben mesylate Structure
Size Price Availability
5mg USD 385 3-4 Weeks
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Quality Control & Documentation
Biological Activity

Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively). Naltriben mesylate displays selectivity for the δ2 subtype in vivo.

Chemical Information
Molecular Weight 511.59
Formula C26H25NO4.CH3SO3H
CAS Number 122517-78-6
Solubility (25°C) DMSO 38 mg/mL (with gentle warming)
Storage -20°C, dry, sealed
References

[1] Thompson, et al. J Pharmacol Exp Ther. VUF10166, a novel compound with differing activities at 5-HT3A and 5-HT3AB receptors.

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Keywords: Naltriben mesylate supplier, TRP Channel, inhibitors, activators

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