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MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors.
| Molecular Weight | 472.67 |
| Formula | C20H20N6S4 |
| CAS Number | 711019-86-2 |
| Solubility (25°C) | DMSO 30 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Geoffrey Burnstock. The therapeutic potential of purinergic signalling
[3] Jiang Bian, et al. P2Y6 Receptor-Mediated Spinal Microglial Activation in Neuropathic Pain
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