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MRS 2279

Cat. No. M7002

All AbMole products are for research use only, cannot be used for human consumption.

MRS 2279 Structure

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Biological Activity

MRS 2279 is a selective, high affinity competitive antagonist of the P2Y1 receptor (Ki = 2.5 nM; IC50 = 51.6 nM). Fails to block nucleotide signaling at most other P2Y receptors (P2Y2, P2Y4, P2Y6, P2Y11 and P2Y12) and potently inhibits ADP-induced aggregation of human blood platelets in vitro (pKB = 8.05).

Chemical Information
Molecular Weight 503.78
Formula C13H18ClN5O8P2.2NH3
CAS Number 367909-40-8
Solubility (25°C) Water 50.38 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Okayama, et al. J Pharmacol Exp Ther. Involvement of concentrative nucleoside transporter 1 in intestinal absorption of trifluorothymidine, a novel antitumor nucleoside, in rats.

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Keywords: MRS 2279 supplier, inhibitors, activators

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