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MLS000545091

Cat. No. M42483

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MLS000545091 Structure

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Quality Control & Documentation
Biological Activity

MLS000545091 is a potent and selective lipoxygenase-2 (LOX-2) inhibitor with an IC50 value of 2.6 μM for h15-LOX-2.

Chemical Information
Molecular Weight 262.73
Formula C14H15ClN2O
CAS Number 322666-76-2
Form Solid
Solubility (25°C) DMSO 20 mg/mL (ultrasonic and warming)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Wan-Chen Tsai et al. Bioorg Med Chem. Kinetic and structural investigations of novel inhibitors of human epithelial 15-lipoxygenase-2

[2] J Brian Jameson 2nd et al. PLoS One. A high throughput screen identifies potent and selective inhibitors to human epithelial 15-lipoxygenase-2

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  Catalog
Abmole Inhibitor Catalog




Keywords: MLS000545091 supplier, Lipoxygenase, inhibitors, activators

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