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Ibutamoren (MK 0677) mesylate is a high affinity ghrelin receptor agonist (pKi = 8.14). Growth hormone (GH) secretagog; stimulates GH release from rat pituitary cells in vitro (EC50 = 1.3 nM) and enhances GH plasma levels in vivo. Also attenuates isoproterenol-induced lipolysis in rat adipocytes in vitro. Orally bioavailable.
| Molecular Weight | 624.77 |
| Formula | C27H36N4O5S.CH3SO3H |
| CAS Number | 159752-10-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 62.48 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related Ghrelin Receptor/GHSR Products |
|---|
| Anamorelin
Anamorelin (RC-1291) is an orally active Ghrelin receptor agonist with an EC50 of 0.74 nM. |
| Capromorelin tartrate
Capromorelin tartrate is a potent ghrelin receptor agonist/growth hormone secretagogue (Ki = 7 nM). |
| JMV 2959
JMV 2959 is a growth hormone secretin receptor type 1A (GHS-R1A) antagonist that acts on LC-PK1 cells and inhibits GHS-R1A with an IC50 value of 32±3 nM. |
| Anamorelin hydrochloride
Anamorelin (RC-1291) hydrochloride is a potent ghrelin receptor agonist with EC50 value of 0.74 nM in the FLIPR assay. |
| AZP-531
AZP-531 is an analogue of unacylated ghrelin designed to improve glycaemic control and reduce weight. |
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